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Suzetrigine, a Non-Opioid Small-Molecule Analgesic: Mechanism of Action, Clinical, and Translational Science.
The discovery and approval of Suzetrigine (VX-548, Journavx) marks a significant breakthrough in pain management. It is the first non-opioid analgesic approved since celecoxib in 1998. Suzetrigine selectively blocks voltage-gated sodium cha…