The S-Nitrosylation of Septin2 (SNO-Septin2) axis: A novel potential therapeutic target for treating aneurysms and dissection.

Drug discoveries & therapeutics 2024 Vol.18(3) p. 207-209

Zhang Y, Qu H, Li C, Li L, He L

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Abstract

Aortic aneurysm and aortic dissection (AAD) are severe life-threatening cardiovascular disorders for which no approved pharmaceutical therapies are currently available. Protein S-nitrosylation (SNO) is a typical redox-dependent posttranslational modification whose role in AAD has yet to be described. Recently, Zhang et al. revealed for the first time that SNO modification of macrophage cytoskeletal protein septin2 promotes vascular inflammation and extracellular matrix degradation in aortic aneurysm. Mechanically, the TIAM1-RAC1(T lymphoma invasion and metastasis-inducing protein 1-Ras-related C3 botulinum toxin substrate 1) axis participates in the progression of AAD induced with S-nitrosylated septin2. More importantly, developing R-ketorolac and NSC23766 compounds that specifically target the TIAM1-RAC1 pathway may be new a potential strategy for alleviating AAD.

추출된 의학 개체 (NER)

유형영어 표현한국어 / 풀이UMLS CUI출처등장
시술 botulinum toxin 보툴리눔독소 주사 dict 1
해부 extracellular matrix scispacy 1
약물 SNO → S-nitrosylation scispacy 1
약물 NSC23766 scispacy 1
질환 aneurysms C0002940
Aneurysm
scispacy 1
질환 Aortic aneurysm C0003486
Aortic Aneurysm
scispacy 1
질환 cardiovascular disorders C0007222
Cardiovascular Diseases
scispacy 1
질환 inflammation C0021368
Inflammation
scispacy 1
질환 TIAM1-RAC1(T lymphoma scispacy 1
질환 lymphoma scispacy 1
기타 Septin2 scispacy 1
기타 SNO-Septin2 scispacy 1
기타 redox-dependent scispacy 1
기타 macrophage cytoskeletal protein septin2 scispacy 1
기타 vascular scispacy 1
기타 metastasis-inducing protein 1-Ras-related C3 botulinum toxin substrate 1 scispacy 1

MeSH Terms

Animals; Humans; Aortic Aneurysm; Aortic Dissection; Molecular Targeted Therapy; Protein Processing, Post-Translational; rac1 GTP-Binding Protein; Septins; Signal Transduction; T-Lymphoma Invasion and Metastasis-inducing Protein 1

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